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Bridging Species for Breakthroughs

Custom-Prepared GPCRs from Any Species, Ready on Demand —
Enhancing Our Extensive Collection of Human and Mouse Receptors.
Contact us for details.

GPCR Catalog

Vast coverage of 550 GPCRs to advance drug discovery

Visit our GPCR Catalog for the complete list of the human and mouse receptors, their concentration-response curves, and more.

250 mouse receptors now available for GPCR research

Our assay platform has added 250 mouse GPCRs to its existing coverage of 300 human GPCRs. Unlock the full potential of drug discovery with our expanded collection of 550 GPCRs.

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Sensitive and all-around

Explore the frontier of drug discovery with our cutting-edge assay platform, featuring GPCR-selective signal amplification technology and unparalleled receptor coverage.

Core business
Panel assays
Technology
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Super-Sensitive GPCR Functional Assays for Accelerated Drug Discovery

550+

GPCRs Available

3 Weeks

Fast Turnaround

~100

Clients Worldwide

Proprietary technology with exceptional sensitivity covering >550 human and mouse GPCRs. Trusted by pharmaceutical, biotech, and academic institutions worldwide.

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Why Choose Tanso Biosciences?

Super-Sensitive

Dramatically amplifies G-protein-dependent signals with exceptional specificity

All-Around Coverage

Works with all GPCRs regardless of coupled Gα proteins or animal species

Potency-Oriented

Measures functional potency, not just binding affinity, in various assay modes

Fast Turnaround

Results delivered in as little as 3 weeks depending on study scope

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Our GPCR Assay Services

FlexPanel48

Focused panels with 48 GPCRs covering 13 therapeutic areas including immunology, oncology, endocrinology, psychiatry, neurology, and more

  • Therapeutic area-specific options
  • Agonist and antagonist modes
  • Customizable

Large-Scale Panels

Comprehensive screening for up to 294 human GPCRs and >250 mouse orthologs

  • Maximum coverage
  • Cross-species comparison
  • Customizable

Safety Panels

Specialized panels to evaluate off-target potency for drug safety assessment

  • Agonist and antagonist modes
  • Customizable

Conc-Dependence Analysis

Detailed dose-response studies in various assay modes

  • Multiple assay modes
  • Flexible study design
  • SAR analysis support

Proprietary GPCR Functional Assay Technology

Our patented technology (WO/2020/026979) delivers remarkable sensitivity and comprehensive coverage for all your GPCR research needs.

Remarkable Sensitivity

Dramatically amplifies G-protein-dependent signals and achieves high signal-to-background ratio

Universal Compatibility

Works with all major Gα proteins (Gq, Gs, Gi/o, G12/13) and cross-species

Multiple Assay Modes

Agonist, antagonist, PAM, NAM modes for comprehensive compound characterization

Proven Validation

99% success rate with 208 out of 210 non-orphan GPCRs tested

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Trusted by Industry Leaders

With nearly 100 clients worldwide, Tanso Biosciences is a trusted partner in GPCR drug discovery for leading pharmaceutical and biotech innovators.

Ken Horne
CEO, Capacity Bio, CA, USA

I highly recommend Tanso Biosciences for their assay platform. Its reliability and industry-leading receptor coverage make it a uniquely valuable guide to GPCR drug discovery. We experienced a quick turnaround time as well.

Researcher
Pharma A

Tanso Bio helps us accelerate structure-activity relationship studies.

Researcher
Pharma B

Tanso Bio's assays have revealed key features of our compounds that would otherwise remain unnoticed.

Sample Reports

Simple 4-Step Process

Request Quotation

Share your study outline and we'll propose experiments. NDA optional.

STEP
1

Place Order

Confirm order, ship compounds to our lab, and make payment.

STEP
2

Wait

The turnaround time can be as short as three weeks, depending on the study scale and design and the backlog of orders.

STEP
3

Receive Report

Get comprehensive study report in PDF format.

STEP
4